Crystal structure of JAK2 JH2-V617F in complex with Bemcentinib
收藏Protein Data Bank Japan2024-11-20 更新2026-04-25 收录
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Crystal structure of JAK2 JH2-V617F in complex with Bemcentinib Descriptor: 1-(3,4-diazatricyclo[9.4.0.0^{2,7}]pentadeca-1(11),2(7),3,5,12,14-hexaen-5-yl)-~{N}3-[(7~{S})-7-pyrrolidin-1-yl-6,7,8,9-tetrahydro-5~{H}-benzo[7]annulen-3-yl]-1,2,4-triazole-3,5-diamine, Tyrosine-protein kinase JAK2 Authors: Haikarainen, T, Silvennoinen, O. Deposit date: 2022-10-11 Release date: 2023-02-01 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Identification of Novel Small Molecule Ligands for JAK2 Pseudokinase Domain. Pharmaceuticals, 16, 2023
创建时间:
2022-10-11



