A Direct Approach to a 6‑Hetarylamino[1,2,4]triazolo[4,3‑<i>b</i>][1,2,4,5]tetrazine Library
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https://figshare.com/articles/dataset/A_Direct_Approach_to_a_6_Hetarylamino_1_2_4_triazolo_4_3_i_b_i_1_2_4_5_tetrazine_Library/2331493
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资源简介：
The
synthesis of 6-hetarylamino[1,2,4]triazolo[4,3-b][1,2,4,5]tetrazines
is reported. The functionalized secondary amines
were constructed via a K2CO3-mediated SNAr reaction of weakly basic hetarylamines with 3-(3,5-dimethylpyrazol-1-yl)[1,2,4]triazolo[4,3-b][1,2,4,5]tetrazines, which allowed displacement 3,5-dimethylpyrazolyl
leaving group. Significantly, the reaction exhibited a broad substrate
scope and proceeded in good yields.
创建时间：
2016-02-18
