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Structural Basis for Cyclic Py-Im Polyamide Allosteric Inhibition of Nuclear Receptor Binding

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Protein Data Bank Japan2024-02-21 更新2026-03-21 收录
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Structural Basis for Cyclic Py-Im Polyamide Allosteric Inhibition of Nuclear Receptor Binding Descriptor: (23R,52R)-23,52-diamino-5,11,17,28,34,40,46,57-octamethyl-2,5,8,11,14,17,20,25,28,31,34,37,40,43,46,49,54,57,60,64-icosaazanonacyclo[54.2.1.1~4,7~.1~10,13~.1~16,19~.1~27,30~.1~33,36~.1~39,42~.1~45,48~]hexahexaconta-1(58),4(66),6,10(65),12,16(64),18,27(63),29,33(62),35,39(61),41,45(60),47,56(59)-hexadecaene-3,9,15,21,26,32,38,44,50,55-decone, 5'-D(*CP*(C38)P*AP*GP*TP*AP*CP*TP*GP*G)-3', CALCIUM ION Authors: Chenoweth, D.M. Deposit date: 2010-08-27 Release date: 2010-09-08 Last modified: 2024-02-21 Method: X-RAY DIFFRACTION (0.95 Å) Cite: Structural basis for cyclic py-im polyamide allosteric inhibition of nuclear receptor binding. J.Am.Chem.Soc., 132, 2010
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2010-08-27
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