Structure of DDR1 receptor tyrosine kinase in complex with inhibitor SR159
收藏Protein Data Bank Japan2024-01-31 更新2026-03-21 收录
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Structure of DDR1 receptor tyrosine kinase in complex with inhibitor SR159 Descriptor: 1,2-ETHANEDIOL, 5-amino-N-(4-(((2S)-4-cyclohexyl-1-((1-(methylsulfonyl)piperidin-3-yl)amino)-1-oxobutan-2-yl)carbamoyl)benzyl)-1-phenyl-1H-pyrazole-4-carboxamide, Epithelial discoidin domain-containing receptor 1, ... Authors: Pinkas, D.M, Bufton, J.C, Roehm, S, Joerger, A.C, Knapp, S, Bullock, A.N, Structural Genomics Consortium (SGC) Deposit date: 2020-12-22 Release date: 2021-03-03 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.87081933411 Å) Cite: Development of a Selective Dual Discoidin Domain Receptor (DDR)/p38 Kinase Chemical Probe. J.Med.Chem., 64, 2021
创建时间:
2020-12-22



