Structure of the mitogen activated kinase kinase 7 in complex with pyrazolopyrimidine 1k
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Structure of the mitogen activated kinase kinase 7 in complex with pyrazolopyrimidine 1k Descriptor: (R)-1-(3-(4-amino-3-(naphthalen-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one, Dual specificity mitogen-activated protein kinase kinase 7 Authors: Wolle, P, Mueller, M.P, Rauh, D. Deposit date: 2019-01-10 Release date: 2019-05-22 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Characterization of Covalent Pyrazolopyrimidine-MKK7 Complexes and a Report on a Unique DFG-in/Leu-in Conformation of Mitogen-Activated Protein Kinase Kinase 7 (MKK7). J.Med.Chem., 62, 2019
创建时间:
2019-01-10



