遇见数据集

p300 KAT domain in complex with KB528

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Protein Data Bank Japan2026-03-04 更新2026-08-24 收录
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p300 KAT domain in complex with KB528 Descriptor: 1,2-ETHANEDIOL, 4-[(2~{S})-1-[[(~{R})-[(3~{S})-7-(1-methylpyrazol-4-yl)-2,3-dihydro-1~{H}-pyrido[2,3-b][1,4]oxazin-3-yl]-phenyl-methyl]amino]propan-2-yl]benzenecarbonitrile, CHLORIDE ION, ... Authors: Rahl, P, Gao, H, Calderon, Y, Wang, Z.-F. Deposit date: 2024-07-19 Release date: 2025-07-23 Last modified: 2026-03-04 Method: X-RAY DIFFRACTION (2 Å) Cite: Catalytic Inhibition of p300 Preferentially Targets IRF4 Oncogenic Activity and Tumor Growth in Multiple Myeloma. Cancer Res., 86, 2026

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2024-07-19
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