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Aminomethyl-Derived Beta Secretase (BACE1) Inhibitors: Engaging Gly230 without an Anilide Functionality

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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Aminomethyl-Derived Beta Secretase (BACE1) Inhibitors: Engaging Gly230 without an Anilide Functionality Descriptor: (4S)-4-[2,4-difluoro-5-({[1-(trifluoromethyl)cyclopropyl]amino}methyl)phenyl]-4-methyl-5,6-dihydro-4H-1,3-thiazin-2-amine, 1,2-ETHANEDIOL, Beta-secretase 1, ... Authors: Parris, K.D, Vajdos, F. Deposit date: 2016-08-22 Release date: 2017-01-11 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.78 Å) Cite: Aminomethyl-Derived Beta Secretase (BACE1) Inhibitors: Engaging Gly230 without an Anilide Functionality. J. Med. Chem., 60, 2017

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2016-08-22
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