Crystal structure of human dihydroorotate dehydrogenase with ML390
收藏Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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Crystal structure of human dihydroorotate dehydrogenase with ML390 Descriptor: 1-DEOXY-1-(7,8-DIMETHYL-2,4-DIOXO-3,4-DIHYDRO-2H-BENZO[G]PTERIDIN-1-ID-10(5H)-YL)-5-O-PHOSPHONATO-D-RIBITOL, ACETATE ION, CHLORIDE ION, ... Authors: Lewis, T.A, Sykes, D.B, Law, J.M, Munoz, B, Scadden, D.T, Rustiguel, J.K, Nonato, M.C, Schreiber, S.L. Deposit date: 2016-05-31 Release date: 2016-10-12 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (1.66 Å) Cite: Development of ML390: A Human DHODH Inhibitor That Induces Differentiation in Acute Myeloid Leukemia. ACS Med Chem Lett, 7, 2016
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2016-05-31



