five

BRD4_BD2_A-1107604

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Protein Data Bank Japan2024-04-03 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5ueu
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资源简介:
BRD4_BD2_A-1107604 Descriptor: Bromodomain-containing protein 4, methyl [(6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetate Authors: Park, C.H. Deposit date: 2017-01-03 Release date: 2017-05-10 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (2.26 Å) Cite: Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors. J. Med. Chem., 60, 2017
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2017-01-03
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