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Mouse fumarylacetoacetate hydrolase complexes with a transition-state mimic of the complete substrate

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Protein Data Bank Japan2023-08-30 更新2026-03-21 收录
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https://pdbj.org/mine/summary/2hzy
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Mouse fumarylacetoacetate hydrolase complexes with a transition-state mimic of the complete substrate Descriptor: 4-(2-CARBOXYETHYL)(HYDROXY)PHOSPHORYL]-3-OXOBUTANOIC ACID, CALCIUM ION, Fumarylacetoacetase, ... Authors: Hurley, T.D, Timm, D.E. Deposit date: 2006-08-09 Release date: 2006-08-22 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (1.35 Å) Cite: Slow-onset inhibition of fumarylacetoacetate hydrolase by phosphinate mimics of the tetrahedral intermediate: kinetics, crystal structure and pharmacokinetics. Biochem.J., 402, 2007
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2006-08-09
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