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Glutamate- and DCKA-bound GluN1/GluN2A agonist binding domains with MPX-007

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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Glutamate- and DCKA-bound GluN1/GluN2A agonist binding domains with MPX-007 Descriptor: 4-hydroxy-5,7-dimethylquinoline-2-carboxylic acid, 5-({[(3,4-difluorophenyl)sulfonyl]amino}methyl)-6-methyl-N-[(2-methyl-1,3-thiazol-5-yl)methyl]pyrazine-2-carboxamide, GLUTAMIC ACID, ... Authors: Mou, T.-C, Sprang, S.R, Hansen, K.B. Deposit date: 2016-05-10 Release date: 2016-09-21 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.72 Å) Cite: Structural Basis for Negative Allosteric Modulation of GluN2A-Containing NMDA Receptors. Neuron, 91, 2016
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2016-05-10
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