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PDK1 in complex with inhibitor MP7

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Protein Data Bank Japan2024-02-21 更新2026-03-21 收录
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PDK1 in complex with inhibitor MP7 Descriptor: 1-(3,4-difluorobenzyl)-2-oxo-N-{(1R)-2-[(2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide, 3-phosphoinositide-dependent protein kinase 1 Authors: Yan, Y, Munshi, S.K, Allison, T. Deposit date: 2010-06-02 Release date: 2010-11-24 Last modified: 2024-02-21 Method: X-RAY DIFFRACTION (1.75 Å) Cite: Genetic and pharmacological inhibition of PDK1 in cancer cells: characterization of a selective allosteric kinase inhibitor. J.Biol.Chem., 286, 2011
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2010-06-02
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