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Aurora B kinase in complex with VX-680

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4b8m
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资源简介:
Aurora B kinase in complex with VX-680 Descriptor: AURORA KINASE B-A, CYCLOPROPANECARBOXYLIC ACID {4-[4-(4-METHYL-PIPERAZIN-1-YL)-6-(5-METHYL-2H-PYRAZOL-3-YLAMINO)-PYRIMIDIN-2-YLSULFANYL]-PHENYL}-AMIDE, INNER CENTROMERE PROTEIN A Authors: Sessa, F, Villa, F. Deposit date: 2012-08-28 Release date: 2013-07-10 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Structural and Biochemical Analysis of an Aurora B Kinase Mutant Reveals a Multistep Activation Mechanism To be Published
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2012-08-28
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