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Tubulin-RB3-TTL in complex with compound SI10

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Protein Data Bank Japan2025-02-19 更新2026-04-19 收录
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https://pdbj.org/mine/summary/8yu9
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Tubulin-RB3-TTL in complex with compound SI10 Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 4-(2-chloranylthieno[3,2-d]pyrimidin-4-yl)-7-methoxy-1,3-dihydroquinoxalin-2-one, CALCIUM ION, ... Authors: Wu, C.Y, Wang, Y.X. Deposit date: 2024-03-27 Release date: 2024-06-05 Last modified: 2025-02-19 Method: X-RAY DIFFRACTION (3.25 Å) Cite: Discovery and mechanistic insights into thieno[3,2-d]pyrimidine and heterocyclic fused pyrimidines inhibitors targeting tubulin for cancer therapy. Eur.J.Med.Chem., 276, 2024
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2024-03-27
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