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Crystal Structure of PAK4 in complex with inhibitor CZH062

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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Crystal Structure of PAK4 in complex with inhibitor CZH062 Descriptor: 2-(4-azanylpiperidin-1-yl)-6-chloranyl-N-(1-methylimidazol-4-yl)quinazolin-4-amine, Serine/threonine-protein kinase PAK 4 Authors: Zhao, F, Li, H. Deposit date: 2017-06-27 Release date: 2018-02-07 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.655 Å) Cite: Structure-Based Design of 6-Chloro-4-aminoquinazoline-2-carboxamide Derivatives as Potent and Selective p21-Activated Kinase 4 (PAK4) Inhibitors. J. Med. Chem., 61, 2018
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2017-06-27
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