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Pa.FabF-C164Q in complex with N-isobutyl-1H-pyrazole-3-carboxamide

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Protein Data Bank Japan2025-05-07 更新2026-04-19 收录
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https://pdbj.org/mine/summary/8cn2
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Pa.FabF-C164Q in complex with N-isobutyl-1H-pyrazole-3-carboxamide Descriptor: 3-oxoacyl-[acyl-carrier-protein] synthase 2, DIMETHYL SULFOXIDE, ~{N}-(2-methylpropyl)-1~{H}-pyrazole-3-carboxamide Authors: Georgiou, C, Brenk, R. Deposit date: 2023-02-21 Release date: 2024-01-10 Last modified: 2025-05-07 Method: X-RAY DIFFRACTION (1.88 Å) Cite: Towards new antibiotics: P. aeruginosa FabF ligands discovered by crystallographic fragment screening followed by hit expansion. Eur.J.Med.Chem., 291, 2025
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2023-02-21
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