five

The MARK3 Kinase Domain Bound To AA-CS-1-008

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Protein Data Bank Japan2024-01-31 更新2026-03-28 收录
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The MARK3 Kinase Domain Bound To AA-CS-1-008 Descriptor: 1,2-ETHANEDIOL, 5-Bromo-4-N-[2-(1H-imidazol-5-yl)ethyl]-2-N-[3-(morpholin-4-ylmethyl)phenyl]pyrimidine-2,4-diamine, MAP/microtubule affinity-regulating kinase 3 Authors: Dederer, V, Preuss, F, Chatterjee, D, Vlassova, A, Mathea, S, Axtman, A, Knapp, S. Deposit date: 2021-07-01 Release date: 2021-07-14 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Identification of Pyrimidine-Based Lead Compounds for Understudied Kinases Implicated in Driving Neurodegeneration. J.Med.Chem., 65, 2022
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2021-07-01
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