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Crystal Structure Matriptase (C731S) in Complex with Inhibitor VD4162B

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Protein Data Bank Japan2024-04-10 更新2026-04-19 收录
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Crystal Structure Matriptase (C731S) in Complex with Inhibitor VD4162B Descriptor: CHLORIDE ION, Cyclic peptide inhibitor (ACE)Y(DTR)(NLE)(KCM), Cyclic peptide inhibitor (ACE)Y(DTR)(NLE)(THZ), ... Authors: Lovell, S, Kashipathy, M.M, Battaile, K.P, Janetka, J.W. Deposit date: 2023-02-03 Release date: 2024-02-07 Last modified: 2024-04-10 Method: X-RAY DIFFRACTION (1.2 Å) Cite: Mechanism-Based Macrocyclic Inhibitors of Serine Proteases. J.Med.Chem., 67, 2024

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2023-02-03
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