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Human p38alpha MAPK in complex with imidazolyl pyridine inhibitor 11b

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5ml5
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资源简介:
Human p38alpha MAPK in complex with imidazolyl pyridine inhibitor 11b Descriptor: 3-(2,5-dimethoxyphenyl)-~{N}-[4-[4-(4-fluorophenyl)-2-methylsulfanyl-1~{H}-imidazol-5-yl]pyridin-2-yl]propanamide, Mitogen-activated protein kinase 14, octyl beta-D-glucopyranoside Authors: Buehrmann, M, Rauh, D. Deposit date: 2016-12-06 Release date: 2017-04-05 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Optimized 4,5-Diarylimidazoles as Potent/Selective Inhibitors of Protein Kinase CK1 delta and Their Structural Relation to p38 alpha MAPK. Molecules, 22, 2017
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2016-12-06
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