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CRYSTAL STRUCTURE OF THE ATPASE REGION OF SACCHAROMYCES CEREVISIAE TOPOISOMERASE II BOUND TO ICRF-187 (DEXRAZOXANE)

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Protein Data Bank Japan2023-08-23 更新2026-03-21 收录
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CRYSTAL STRUCTURE OF THE ATPASE REGION OF SACCHAROMYCES CEREVISIAE TOPOISOMERASE II BOUND TO ICRF-187 (DEXRAZOXANE) Descriptor: (S)-4,4'-(1-METHYL-1,2-ETHANEDIYL)BIS-2,6-PIPERAZINEDIONE, DNA topoisomerase II, MAGNESIUM ION, ... Authors: Classen, S, Olland, S, Berger, J.M. Deposit date: 2003-09-17 Release date: 2003-09-30 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Structure of the topoisomerase II ATPase region and its mechanism of inhibition by the chemotherapeutic agent ICRF-187 Proc.Natl.Acad.Sci.USA, 100, 2003

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2003-09-17
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