POLYADPRIBOSYL GLYCOSIDASE IN COMPLEX WITH PDD00017262
收藏Protein Data Bank Japan2025-08-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5lhb
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POLYADPRIBOSYL GLYCOSIDASE IN COMPLEX WITH PDD00017262 Descriptor: 1-(cyclopropylmethyl)-6-[[(1-methylcyclopropyl)amino]-bis(oxidanyl)-$l^{4}-sulfanyl]-3-[(2-methyl-1,3-thiazol-5-yl)methyl]quinazoline-2,4-dione, DIMETHYL SULFOXIDE, Poly(ADP-ribose) glycohydrolase, ... Authors: Tucker, J, Barkauskaite, E. Deposit date: 2016-07-10 Release date: 2016-10-12 Last modified: 2025-08-06 Method: X-RAY DIFFRACTION (2.23 Å) Cite: First-in-Class Chemical Probes against Poly(ADP-ribose) Glycohydrolase (PARG) Inhibit DNA Repair with Differential Pharmacology to Olaparib. ACS Chem. Biol., 11, 2016
创建时间:
2016-07-10



