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MerTK kinase domain in complex with purine inhibitor

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Protein Data Bank Japan2024-05-01 更新2026-03-21 收录
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https://pdbj.org/mine/summary/7aw0
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资源简介:
MerTK kinase domain in complex with purine inhibitor Descriptor: 2-(cyclopentyloxy)-9-(2,6-difluorobenzyl)-N-methyl-9H-purin-6-amine, Tyrosine-protein kinase Mer Authors: Schimpl, M, Nissink, J.W.M, Blackett, C, Clarke, M, Disch, J, Goldberg, K, Guilinger, J, Hennessy, E.J, Jetson, R, Ginkunja, D, Hardaker, E, Keefe, A, McCoull, W, McMurray, L, Collingwood, O, Overman, R, Pflug, A, Preston, M, Rawlins, P, Rivers, E, Smith, P, Underwood, E, Truman, C, Warwicker, J, Winter, J, Woodcock, S, Zhang, Y. Deposit date: 2020-11-06 Release date: 2021-03-03 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (1.893 Å) Cite: Generating Selective Leads for Mer Kinase Inhibitors-Example of a Comprehensive Lead-Generation Strategy. J.Med.Chem., 64, 2021
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2020-11-06
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