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Complex of the phosphorylated human cystic fibrosis transmembrane conductance regulator (CFTR) with CFTRinh-172 and ATP/Mg

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Protein Data Bank Japan2024-03-20 更新2026-06-30 收录
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https://pdbj.org/mine/summary/8ubr
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Complex of the phosphorylated human cystic fibrosis transmembrane conductance regulator (CFTR) with CFTRinh-172 and ATP/Mg Descriptor: 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine, 4-[(Z)-{(3M)-4-oxo-2-sulfanylidene-3-[3-(trifluoromethyl)phenyl]-1,3-thiazolidin-5-ylidene}methyl]benzoic acid, ADENOSINE-5'-TRIPHOSPHATE, ... Authors: Young, P.G, Fiedorczuk, K, Chen, J. Deposit date: 2023-09-24 Release date: 2024-02-21 Last modified: 2024-03-20 Method: ELECTRON MICROSCOPY (2.7 Å) Cite: Structural basis for CFTR inhibition by CFTR inh -172. Proc.Natl.Acad.Sci.USA, 121, 2024
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2023-09-24
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