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CRYSTAL STRUCTURE OF HUMAN TANKYRASE-2 IN COMPLEX WITH A PYRANOPYRIDONE INHIBITOR

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Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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CRYSTAL STRUCTURE OF HUMAN TANKYRASE-2 IN COMPLEX WITH A PYRANOPYRIDONE INHIBITOR Descriptor: (3R)-3-(1-hydroxy-2-methylpropan-2-yl)-1,3,4,5-tetrahydro-6H-pyrano[4,3-c]isoquinolin-6-one, SULFATE ION, Tankyrase-2, ... Authors: Lukacs, C.M, Janson, C.A. Deposit date: 2015-06-21 Release date: 2015-08-12 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (1.75 Å) Cite: Fragment-Based Drug Design of Novel Pyranopyridones as Cell Active and Orally Bioavailable Tankyrase Inhibitors. Acs Med.Chem.Lett., 6, 2015
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2015-06-21
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