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crystal structure of HIV model protease precursor/saquinavir complex

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Protein Data Bank Japan2023-09-13 更新2026-03-21 收录
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crystal structure of HIV model protease precursor/saquinavir complex Descriptor: (2S)-N-[(2S,3R)-4-[(2S,3S,4aS,8aS)-3-(tert-butylcarbamoyl)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-hydroxy-1 -phenyl-butan-2-yl]-2-(quinolin-2-ylcarbonylamino)butanediamide, CHLORIDE ION, GLYCEROL, ... Authors: Agniswamy, J, Sayer, J, Weber, I, Louis, J. Deposit date: 2011-08-26 Release date: 2012-04-25 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (1.36 Å) Cite: Terminal interface conformations modulate dimer stability prior to amino terminal autoprocessing of HIV-1 protease. Biochemistry, 51, 2012

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2011-08-26
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