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InhA in complex with a DNA encoded library hit

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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InhA in complex with a DNA encoded library hit Descriptor: 5-[(4-fluoranyl-3-phenoxy-phenyl)methylamino]-~{N}-methyl-6-[(1-pyridin-2-ylpiperidin-4-yl)amino]pyridine-3-carboxamide, ENOYL-[ACYL-CARRIER-PROTEIN] REDUCTASE [NADH], NICOTINAMIDE-ADENINE-DINUCLEOTIDE Authors: Read, J.A, Breed, J. Deposit date: 2016-03-22 Release date: 2016-11-30 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (1.73 Å) Cite: Discovery of Cofactor-Specific, Bactericidal Mycobacterium Tuberculosis Inha Inhibitors Using DNA-Encoded Library Technology Proc.Natl.Acad.Sci.USA, 113, 2016

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2016-03-22
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