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HUMAN PFKFB3 IN COMPLEX WITH KAN0438241

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Protein Data Bank Japan2025-04-09 更新2026-03-21 收录
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HUMAN PFKFB3 IN COMPLEX WITH KAN0438241 Descriptor: 4-[[3-(5-fluoranyl-2-oxidanyl-phenyl)phenyl]sulfonylamino]-2-oxidanyl-benzoic acid, 6-O-phosphono-beta-D-fructofuranose, 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3, ... Authors: Gustafsson, N.M.S, Lundback, T, Farnegardh, K, Groth, P, Wiitta, E, Jonsson, M, Hallberg, K, Pennisi, R, Huguet Ninou, A, Martinsson, J, Norstrom, C, Schultz, J, Andersson, M, Markova, N, Marttila, P, Norin, M, Olin, T, Helleday, T. Deposit date: 2017-10-26 Release date: 2018-11-07 Last modified: 2025-04-09 Method: X-RAY DIFFRACTION (2.51 Å) Cite: Targeting PFKFB3 radiosensitizes cancer cells and suppresses homologous recombination. Nat Commun, 9, 2018
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2017-10-26
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