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Focal Adhesion Kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/2jko
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Focal Adhesion Kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor Descriptor: 7-{[(2Z,5S)-5-CHLORO-2-{[2-METHOXY-4-(4-METHYLPIPERAZIN-1-YL)PHENYL]IMINO}-2,5-DIHYDROPYRIMIDIN-4-YL]AMINO}-2-METHYL-2,3-DIHYDRO-1H-ISOINDOL-1-ONE, FOCAL ADHESION KINASE 1 Authors: Lietha, D, Eck, M.J. Deposit date: 2008-08-28 Release date: 2008-09-09 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (1.65 Å) Cite: Crystal Structures of the Fak Kinase in Complex with Tae226 and Related Bis-Anilino Pyrimidine Inhibitors Reveal a Helical Dfg Conformation. Plos One, 3, 2008
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2008-08-28
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