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Crystal structures of JAK1 and JAK2 inhibitor complexes

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Protein Data Bank Japan2024-11-27 更新2026-03-21 收录
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Crystal structures of JAK1 and JAK2 inhibitor complexes Descriptor: 3-{(3R,4R)-4-methyl-3-[methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile, Tyrosine-protein kinase JAK2 Authors: Williams, N.K, Bamert, R.S, Patel, O, Fantino, E, Rossjohn, J, Lucet, I.S. Deposit date: 2009-01-14 Release date: 2009-02-10 Last modified: 2024-11-27 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Dissecting specificity in the Janus kinases: the structures of JAK-specific inhibitors complexed to the JAK1 and JAK2 protein tyrosine kinase domains. J.Mol.Biol., 387, 2009

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2009-01-14
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