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Crystal structure of human ATAD2 bromodomain in complex with N-(4-bromo-3-(3-methylpyrrolidin-1-yl)sulfonyl)phenyl)-2-(-4-cyclopropyl-4-methyl-2,5-dioxoimidazolidin-1-yl)acetamide

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Protein Data Bank Japan2024-05-15 更新2026-03-21 收录
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Crystal structure of human ATAD2 bromodomain in complex with N-(4-bromo-3-(3-methylpyrrolidin-1-yl)sulfonyl)phenyl)-2-(-4-cyclopropyl-4-methyl-2,5-dioxoimidazolidin-1-yl)acetamide Descriptor: 1,2-ETHANEDIOL, ATPase family AAA domain-containing protein 2, SULFATE ION, ... Authors: Chung, C. Deposit date: 2020-03-15 Release date: 2020-05-06 Last modified: 2024-05-15 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Optimization of Potent ATAD2 and CECR2 Bromodomain Inhibitors with an Atypical Binding Mode. J.Med.Chem., 63, 2020
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2020-03-15
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