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Crystal structure of the ATP binding domain of S. aureus GyrB complexed with a fragment

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Protein Data Bank Japan2024-12-25 更新2026-03-21 收录
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Crystal structure of the ATP binding domain of S. aureus GyrB complexed with a fragment Descriptor: (4S)-2-METHYL-2,4-PENTANEDIOL, 5-(thiophen-2-yl)thieno[2,3-d]pyrimidin-4(1H)-one, CHLORIDE ION, ... Authors: Andersen, O.A, Barker, J, Cheng, R.K, Kahmann, J, Felicetti, B, Wood, M, Scheich, C, Mesleh, M, Cross, J.B, Zhang, J, Yang, Q, Lippa, B, Ryan, M.D. Deposit date: 2015-07-24 Release date: 2016-02-03 Last modified: 2024-12-25 Method: X-RAY DIFFRACTION (1.45 Å) Cite: Fragment-based discovery of DNA gyrase inhibitors targeting the ATPase subunit of GyrB. Bioorg.Med.Chem.Lett., 26, 2016
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2015-07-24
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