ABCG2 topotecan turnover-1 state
收藏Protein Data Bank Japan2024-10-16 更新2026-03-28 收录
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ABCG2 topotecan turnover-1 state Descriptor: (S)-10-[(DIMETHYLAMINO)METHYL]-4-ETHYL-4,9-DIHYDROXY-1H-PYRANO[3',4':6,7]INOLIZINO[1,2-B]-QUINOLINE-3,14(4H,12H)-DIONE, ADENOSINE-5'-TRIPHOSPHATE, Broad substrate specificity ATP-binding cassette transporter ABCG2, ... Authors: Yu, Q, Ni, D, Kowal, J, Manolaridis, I, Jackson, S.M, Stahlberg, H, Locher, K.P. Deposit date: 2021-05-15 Release date: 2021-07-21 Last modified: 2024-10-16 Method: ELECTRON MICROSCOPY (3.1 Å) Cite: Structures of ABCG2 under turnover conditions reveal a key step in the drug transport mechanism. Nat Commun, 12, 2021
创建时间:
2021-05-15



