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SETD7 in complex with inhibitor PF-5426 and S-adenosyl-methionine

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Protein Data Bank Japan2023-09-20 更新2026-03-21 收录
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SETD7 in complex with inhibitor PF-5426 and S-adenosyl-methionine Descriptor: Histone-lysine N-methyltransferase SETD7, N-[(2R)-3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-8-fluoro-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide, S-ADENOSYLMETHIONINE, ... Authors: Dong, A, Wu, H, Zeng, H, Park, H, El Bakkouri, M, Barsyte, D, Vedadi, M, Tatlock, J, Owen, D, Bunnage, M, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Brown, P.J, Structural Genomics Consortium (SGC) Deposit date: 2013-02-25 Release date: 2013-03-27 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (1.7 Å) Cite: SETD7 in complex with inhibitor PF-5426 and S-adenosyl-methionine to be published
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2013-02-25
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