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Crystal structure of Lp-PLA2 in complex with a novel covalent inhibitor

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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Crystal structure of Lp-PLA2 in complex with a novel covalent inhibitor Descriptor: (2S)-2-[(Z)-1,3-bis(oxidanyl)-3-oxidanylidene-prop-1-enyl]pyrrolidine-1-carboxylic acid, Platelet-activating factor acetylhydrolase Authors: Hu, H.C, Xu, Y.C. Deposit date: 2020-02-20 Release date: 2020-12-30 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Identification of Highly Selective Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Inhibitors by a Covalent Fragment-Based Approach. J.Med.Chem., 63, 2020
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2020-02-20
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