C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH GSK620
收藏Protein Data Bank Japan2024-05-01 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6zb1
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C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH GSK620 Descriptor: 1,2-ETHANEDIOL, Bromodomain-containing protein 2, ~{N}5-cyclopropyl-~{N}3-methyl-2-oxidanylidene-1-(phenylmethyl)pyridine-3,5-dicarboxamide Authors: Chung, C. Deposit date: 2020-06-06 Release date: 2020-08-05 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (1.6 Å) Cite: The Optimization of a Novel, Weak Bromo and Extra Terminal Domain (BET) Bromodomain Fragment Ligand to a Potent and Selective Second Bromodomain (BD2) Inhibitor. J.Med.Chem., 63, 2020
创建时间:
2020-06-06



