Crystal structure of human BCL6 BTB domain in complex with compound 23d
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Crystal structure of human BCL6 BTB domain in complex with compound 23d Descriptor: 1,2-ETHANEDIOL, 5-[[5-chloranyl-2-(3,5-dimethylpyrazol-1-yl)pyrimidin-4-yl]amino]-1-methyl-3-(3-methyl-3-oxidanyl-butyl)benzimidazol-2-one, ALA-TRP-VAL-ILE-PRO-ALA, ... Authors: Rodrigues, M.J, Le Bihan, Y.-V, van Montfort, R.L.M. Deposit date: 2019-12-11 Release date: 2020-04-22 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.43 Å) Cite: AchievingIn VivoTarget Depletion through the Discovery and Optimization of Benzimidazolone BCL6 Degraders. J.Med.Chem., 63, 2020
创建时间:
2019-12-11



