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Protein kinase A mutants as surrogate model for Aurora B with AT9283 inhibitor

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5n23
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Protein kinase A mutants as surrogate model for Aurora B with AT9283 inhibitor Descriptor: 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1H-benzimidazol-2-yl]-1H-pyrazol-4-yl}urea, cAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase inhibitor alpha Authors: Alam, K.A, Rothweiler, U, Engh, R.A. Deposit date: 2017-02-07 Release date: 2018-03-14 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.088 Å) Cite: Inhibitor induced structural effects involving Phe327 in AGC kinases To Be Published
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2017-02-07
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