HDAC6 selective degraded (difluoromethyl)-1,3,4-oxadiazole substrate inhibitor
收藏Protein Data Bank Japan2023-11-01 更新2026-04-25 收录
下载链接:
https://pdbj.org/mine/summary/8cj7
下载链接
链接失效反馈官方服务:
资源简介:
HDAC6 selective degraded (difluoromethyl)-1,3,4-oxadiazole substrate inhibitor Descriptor: 6-[(5-pyridin-2-yl-1,2$l^{4},3,4-tetrazacyclopenta-1,3-dien-2-yl)methyl]pyridine-3-carbohydrazide, Histone deacetylase 6, IODIDE ION, ... Authors: Sandmark, J, Ek, M, Ripa, L. Deposit date: 2023-02-12 Release date: 2023-10-18 Last modified: 2023-11-01 Method: X-RAY DIFFRACTION (1.51 Å) Cite: Selective and Bioavailable HDAC6 2-(Difluoromethyl)-1,3,4-oxadiazole Substrate Inhibitors and Modeling of Their Bioactivation Mechanism. J.Med.Chem., 66, 2023
创建时间:
2023-02-12



