RORgamma in complex with inverse agonist BIO399.
收藏Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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RORgamma in complex with inverse agonist BIO399. Descriptor: N-(5-ethyl-3,3-dimethyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-8-yl)-3,4-dimethyl-N-(2,2,2-trifluoroethyl)benzene-1-sulfonamide, Nuclear receptor ROR-gamma Authors: Marcotte, D.J. Deposit date: 2016-03-23 Release date: 2016-06-15 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (2.35 Å) Cite: Structural determinant for inducing RORgamma specific inverse agonism triggered by a synthetic benzoxazinone ligand. Bmc Struct.Biol., 16, 2016
创建时间:
2016-03-23



