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Crystal Structure of PAK4 in complex with inhibitor CZH216

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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Crystal Structure of PAK4 in complex with inhibitor CZH216 Descriptor: ETHANOL, Serine/threonine-protein kinase PAK 4, [6-chloranyl-4-[(5-methyl-1H-pyrazol-3-yl)amino]quinazolin-2-yl]-[(3R)-3-methylpiperazin-1-yl]methanone Authors: Zhao, F, Li, H. Deposit date: 2017-06-27 Release date: 2018-02-07 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (1.847 Å) Cite: Structure-Based Design of 6-Chloro-4-aminoquinazoline-2-carboxamide Derivatives as Potent and Selective p21-Activated Kinase 4 (PAK4) Inhibitors. J. Med. Chem., 61, 2018
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2017-06-27
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