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Crystal structure of P21-activated kinase 1 in complex with an inhibitor compound 29

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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Crystal structure of P21-activated kinase 1 in complex with an inhibitor compound 29 Descriptor: N~2~-[(7-chloro-1H-benzimidazol-6-yl)methyl]-N~4~-(5-cyclopropyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine, SULFATE ION, Serine/threonine-protein kinase PAK 1 Authors: Rouge, L, Wang, W. Deposit date: 2015-05-21 Release date: 2015-07-01 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.15 Å) Cite: Structure-Guided Design of Group I Selective p21-Activated Kinase Inhibitors. J.Med.Chem., 58, 2015
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2015-05-21
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