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Notum Inhibitor ARUK3005522

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Protein Data Bank Japan2024-11-13 更新2026-04-19 收录
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Notum Inhibitor ARUK3005522 Descriptor: (3~{a}~{R})-2,3,3~{a},4-tetrahydropyrrolo[1,2-a]indol-1-one, 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... Authors: Zhao, Y, Jones, E.Y, Fish, P. Deposit date: 2022-11-27 Release date: 2022-12-14 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.7 Å) Cite: Designed switch from covalent to non-covalent inhibitors of carboxylesterase Notum activity. Eur.J.Med.Chem., 251, 2023

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2022-11-27
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