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Three-Dimensional Structure of Human Carbonic Anhydrase IX in Complex with a Covalent Inhibitor

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Protein Data Bank Japan2025-01-22 更新2026-04-19 收录
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Three-Dimensional Structure of Human Carbonic Anhydrase IX in Complex with a Covalent Inhibitor Descriptor: 3-[[(1~{R},4~{Z})-cyclododec-4-en-1-yl]amino]-4-ethylsulfonyl-2,5,6-tris(fluoranyl)benzenesulfonamide, Carbonic anhydrase, ZINC ION Authors: Leitans, J, Tars, K. Deposit date: 2024-06-05 Release date: 2024-12-18 Last modified: 2025-01-22 Method: X-RAY DIFFRACTION (2.2 Å) Cite: Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX. Elife, 13, 2024

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2024-06-05
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