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Protein farnesyltransferase complexed with FPP and ethylenediamine scaffold inhibitor 2

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Protein Data Bank Japan2024-02-21 更新2026-03-21 收录
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https://pdbj.org/mine/summary/3e32
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Protein farnesyltransferase complexed with FPP and ethylenediamine scaffold inhibitor 2 Descriptor: FARNESYL DIPHOSPHATE, N-benzyl-N-(2-{(4-cyanophenyl)[(1-methyl-1H-imidazol-5-yl)methyl]amino}ethyl)-1-methyl-1H-imidazole-4-sulfonamide, Protein farnesyltransferase subunit beta, ... Authors: Hast, M.A, Beese, L.S. Deposit date: 2008-08-06 Release date: 2009-03-10 Last modified: 2024-02-21 Method: X-RAY DIFFRACTION (2.45 Å) Cite: Structural basis for binding and selectivity of antimalarial and anticancer ethylenediamine inhibitors to protein farnesyltransferase. Chem.Biol., 16, 2009
创建时间:
2008-08-06
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