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Crystal structure of the human alpha1B adrenergic receptor in complex with inverse agonist (+)-cyclazosin

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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https://pdbj.org/mine/summary/7b6w
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Crystal structure of the human alpha1B adrenergic receptor in complex with inverse agonist (+)-cyclazosin Descriptor: Alpha-1B adrenergic receptor,alpha1B adrenergic receptor,Alpha-1B adrenergic receptor,alpha1B adrenergic receptor,Alpha-1B adrenergic receptor,alpha1B adrenergic receptor,Alpha-1B adrenergic receptor,alpha1B adrenergic receptor, [(4~{a}~{R},8~{a}~{S})-4-(4-azanyl-6,7-dimethoxy-quinazolin-2-yl)-2,3,4~{a},5,6,7,8,8~{a}-octahydroquinoxalin-1-yl]-(furan-2-yl)methanone Authors: Deluigi, M, Morstein, L, Hilge, M, Schuster, M, Merklinger, L, Klipp, A, Scott, D.J, Plueckthun, A. Deposit date: 2020-12-08 Release date: 2022-01-12 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.873 Å) Cite: Crystal structure of the alpha 1B -adrenergic receptor reveals molecular determinants of selective ligand recognition. Nat Commun, 13, 2022
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2020-12-08
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