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Bromodomain-containing 4 BD1 in complex with 3',4',7,8-Tetrahydroxyflavone

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Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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https://pdbj.org/mine/summary/7c2z
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资源简介:
Bromodomain-containing 4 BD1 in complex with 3',4',7,8-Tetrahydroxyflavone Descriptor: 2-[3,4-bis(oxidanyl)phenyl]-7,8-bis(oxidanyl)chromen-4-one, Bromodomain-containing protein 4, FORMIC ACID Authors: Li, J, Zhu, J. Deposit date: 2020-05-10 Release date: 2021-05-12 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (1.3 Å) Cite: Discovery of the natural product 3',4',7,8-tetrahydroxyflavone as a novel and potent selective BRD4 bromodomain 2 inhibitor. J Enzyme Inhib Med Chem, 36, 2021
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2020-05-10
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