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FGFR2 kinase domain with a macrocyclic compound 8g

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Protein Data Bank Japan2026-02-04 更新2026-04-19 收录
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https://pdbj.org/mine/summary/9u7e
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资源简介:
FGFR2 kinase domain with a macrocyclic compound 8g Descriptor: (E)-4-methyl-17-(1-methyl-1H-pyrazol-4-yl)-7,10-dioxa-4-aza-1(3,6)-imidazo[1,2-b]pyridazina-2(3,5)-pyridinacyclodecaphan-3-one, Fibroblast growth factor receptor 2, SULFATE ION Authors: Chen, X.J, Chen, Y.H. Deposit date: 2025-03-24 Release date: 2026-01-21 Last modified: 2026-02-04 Method: X-RAY DIFFRACTION (2.2 Å) Cite: Design, Synthesis, and Biological Evaluation of the First Novel Macrocycle-Based FGFR Inhibitors That Overcome Clinically Acquired Resistance. J.Med.Chem., 69, 2026
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2025-03-24
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