Ash1L SET domain in complex with AS-85
收藏Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6wzw
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资源简介：
Ash1L SET domain in complex with AS-85 Descriptor: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Histone-lysine N-methyltransferase ASH1L, N-{[3-(3-carbamothioylphenyl)-1-{1-[(trifluoromethyl)sulfonyl]piperidin-4-yl}-1H-indol-6-yl]methyl}azetidine-3-carboxamide, ... Authors: Li, H, Deng, J, Cierpicki, T, Grembecka, J. Deposit date: 2020-05-14 Release date: 2021-04-07 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.69 Å) Cite: Discovery of first-in-class inhibitors of ASH1L histone methyltransferase with anti-leukemic activity. Nat Commun, 12, 2021
创建时间：
2020-05-14
