Crystal structure of the bromodomain of human CREBBP bound to the benzodiazepinone G02857790
收藏Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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Crystal structure of the bromodomain of human CREBBP bound to the benzodiazepinone G02857790 Descriptor: (4R)-6-(3-cyclopropyl-1-methyl-1H-indazol-5-yl)-4-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-2-one, ACETATE ION, CALCIUM ION, ... Authors: Setser, J.W, Poy, F, Bellon, S.F. Deposit date: 2016-02-18 Release date: 2016-04-20 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (1.07 Å) Cite: Fragment-Based Discovery of a Selective and Cell-Active Benzodiazepinone CBP/EP300 Bromodomain Inhibitor (CPI-637). Acs Med.Chem.Lett., 7, 2016
创建时间：
2016-02-18
