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Isolated p110a subunit of PI3Ka provides a platform for structure-based drug design

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Protein Data Bank Japan2023-12-27 更新2026-03-21 收录
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Isolated p110a subunit of PI3Ka provides a platform for structure-based drug design Descriptor: 2-amino-8-[trans-4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8H)-one, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform Authors: Chen, P, Deng, Y.-L, Bergqvist, S, Falk, M, Liu, W, Timofeevski, S. Deposit date: 2014-06-25 Release date: 2014-08-06 Last modified: 2023-12-27 Method: X-RAY DIFFRACTION (2.85 Å) Cite: Engineering of an isolated p110 alpha subunit of PI3K alpha permits crystallization and provides a platform for structure-based drug design. Protein Sci., 23, 2014
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2014-06-25
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